adenosine receptor — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T14127	Adenosine A1 receptor activator T62		Adenosine Receptor
	Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor, and it produces antinociception in animal models of acute pain and also reduces hypersensitivity in models of inflammatory and nerve...		Adenosine Receptor
T22466	Adenosine receptor A1 antagonist 5		cAMP
	Adenosine receptor A1 antagonist 5 acts as an adenosine antagonist, is an oxypurine, acts as an insecticide and pest control agent, and has an inhibitory effect on elevated blood pressure.		cAMP
T21620	Adenosine receptor antagonist 4		Adenosine Receptor
	Adenosine receptor antagonist 4 is an adenosine receptor antagonist.		Adenosine Receptor
T40307	Adenosine receptor antagonist 1
	Adenosine receptor antagonist 1 is a highly selective antagonist for the A2aR adenosine receptor, exhibiting an IC50 value of 0.29 nM. It demonstrates a remarkable 14-fold selectivity towards the A2aR receptor in compari...
T7683	Adenosine amine congener	ADAC	Adenosine Receptor
	Adenosine amine congener (ADAC) (ADAC) is an agonist of selective A1 adenosine receptor,.		Adenosine Receptor
T12163	N6-(2-Phenylethyl)adenosine	N6-Phenethyladenosine,N6-Phenylethyladenosine	Adenosine Receptor
	N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine) is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM for rat and human A1.		Adenosine Receptor
TN2247	Swertisin		Adenosine Receptor
	Swertisin, a novel herbal biomolecule, shows a strong antihyperglycemic action. Swertisin is an adenosine A1 receptor antagonist, is known to have antidiabetic, anti-inflammatory and antioxidant effects.		Adenosine Receptor
T22234	Alloxazine		Adenosine Receptor
	Alloxazine (Isoalloxazine) is an A2 receptor antagonist, which is approximately 10-fold more selective for the A2B receptor than for the A2A receptor.		Adenosine Receptor
T16136	MRS-1706		Adenosine Receptor
	MRS-1706 has Ki values of 1.39, 112, 157, and 230 nM for human A2B, A2A, A1, and A3 receptors respectively. MRS-1706 is an effective and selective adenosine A2B receptor inverse agonist.		Adenosine Receptor
T0853L	Adenosine 5'-monophosphate monohydrate	5'-AMP,5'-AMP monohydrate,5'-Adenylic acid	AMPK , Adenosine Receptor , HSV
	Adenosine 5'-monophosphate monohydrate (5'-AMP) , also known as 5'-adenylic acid, is a nucleotide that is used as a monomer in RNA. It is an ester of phosphoric acid and the nucleoside adenosine. Adenosine 5'-monophospha...		AMPK , Adenosine Receptor , HSV
T12164	N6-(4-Hydroxybenzyl)adenosine	Para-topolin riboside	P2Y Receptor
	N6-(4-Hydroxybenzyl)adenosine (Para-topolin riboside) is a platelet aggregation inhibitor.		P2Y Receptor
T8551	Nitrobenzylthioinosine	NBMPR	AChR , Adenosine Receptor
	Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.		AChR , Adenosine Receptor
T12161	N6-Ethyladenosine		Adenosine Receptor
	N6-Ethyladenosine is an adenosine derivative, acts as an agonist of Adenosine receptor(hA1AR and hA3AR with Kis of 4.9 and 4.7 nM , respectively).		Adenosine Receptor
T8512	BAY-545		Adenosine Receptor
	BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).		Adenosine Receptor
T14078	AB928		Adenosine Receptor
	AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].		Adenosine Receptor
T16140	MRS 1754		Adenosine Receptor
	MRS 1754 is a selective antagonist radioligand for the A2B adenosine receptor. It has a very low affinity for A1 and A3 receptors of both humans and rats.		Adenosine Receptor
T7021	ZM241385		Adenosine Receptor
	ZM-241385 is a high-affinity antagonist ligand selective for the adenosine A2A receptor.		Adenosine Receptor
T1681	Aminophylline	Phyllocontin	PDE , Adenosine Receptor
	Aminophylline (Phyllocontin) is a competitive nonselective phosphodiesterase inhibitor giving a bronchodilatory effect.		PDE , Adenosine Receptor
T8312	Derenofylline		Adenosine Receptor
	Derenofylline is a selective and potent adenosine A(1) antagonist in vitro (Ki=1 nM)		Adenosine Receptor
T6979	SCH 58261	SCH58261	Adenosine Receptor
	SCH 58261 is a potent and selective A2a adenosine receptor antagonist.The Ki =2.3 nM for rat A2a and 2 nM is for bovine A2a.		Adenosine Receptor